Product Name | Brefeldin A (Synonyms: BFA ; Cyanein ; Decumbin) |
---|---|
CAS | 20350-15-6 |
Formula | C16H24O4 |
MW | 280.36 |
MDL | MFCD00083258 |
Appearance | Off-white powder |
Storage condition | Dry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years). |
Brefeldin A (BFA) is a lactone antibiotic and ATPase inhibitor for protein transport with IC50 of 0.2 μM in HCT 116 cells, induces cancer cell differentiation and apoptosis. It could also improve the HDR(homology-directed repair) efficiency and be an enhancer of CRISPR-mediated HDR. Brefeldin A is also an inhibitor of autophagy and mitophagy.
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