拉格鲁西布二盐酸盐 | CHIR-99021二盐酸盐 |
Laduviglusib dihydrochloride | CHIR-99021 dihydrochloride | CT99021 dihydrochloride
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Product Name Laduviglusib dihydrochloride | CHIR-99021 dihydrochloride | CT99021 dihydrochloride
CAS2109414-84-6
FormulaC22H18Cl2N8·2HCl
MW538.26
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Laduviglusib (CHIR-99021) dihydrochloride is a potent and selective GSK-3α/β inhibitor with IC50s of 10 nM and 6.7 nM. Laduviglusib monohydrochloride shows >500-fold selectivity for GSK-3 over CDC2, ERK2 and other protein kinases. Laduviglusib monohydrochloride is also a potent Wnt/β-catenin signaling pathway activator. Laduviglusib monohydrochloride enhances mouse and human embryonic stem cells self-renewal. Laduviglusib monohydrochloride induces autophagy.


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Related
Laduviglusib trihydrochloride | CHIR-99021 Trihydrochloride
Laduviglusib monohydrochloride | CHIR-99021 Monohydrochloride | T99021 Monohydrochloride
Laduviglusib (Synonyms: CHIR-99021; CT99021)
History
Urelumab (Anti-TNFRSF9 / 4-1BB / CD137)
Laduviglusib dihydrochloride | CHIR-99021 dihydrochloride | CT99021 dihydrochloride
Alexa fluor 647 NHS ester
trans-Doxercalciferol