替沃扎尼
Tivozanib (AV-951)
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Product Overview
Product Name Tivozanib (AV-951)
CAS475108-18-0
FormulaC22H19ClN4O5
MW454.86
AppearanceLight brown to brown powder
Storage conditionDry, dark and at 0 - 4℃ for short term (days to weeks) or -20℃ for long term (months to years).
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Product details

Tivozanib is a potent and selective VEGFR inhibitor for VEGFR1/2/3 with IC50 of 30 nM/6.5 nM/15 nM, and also inhibits PDGFR and c-Kit, low activity observed against FGFR-1, Flt3, c-Met, EGFR and IGF-1R. Phase 3.

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History
A-1331852
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