GS-9973| Entospletinib
Entospletinib | GS-9973
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5 mg 10 mg
Product Availability
3-5days
Price
$88.00
Member price
Product Availability
3-5days
Price
$146.00
Member price
Quantity
- +
Product Overview
Product Name Entospletinib | GS-9973
CAS1229208-44-9
FormulaC23H21N7O
MW411.46
AppearanceWhite to gray powder
Storage conditionStore in a dry and dark sealed container, short-term (weeks to months) storage at 0-4 ℃, long-term (months to years) storage at -20 ℃.
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Product details

Entospletinib (GS-9973) is an orally bioavailable, selective Syk inhibitor with IC50 of 7.7 nM in a cell-free assay and showed 13- to >1000-fold cellular selectivity for Syk over other kinases(including Jak2, ckit, Flt3, Ret, KDR) as assessed by target protein phosphorylation or functional response.

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History
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