Olcegepant hydrochloride (BIBN-4096 hydrochloride; BIBN4096BS hydrochloride)
Olcegepant hydrochloride (Synonyms: BIBN-4096 hydrochloride; BIBN4096BS hydrochloride)
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Product Name Olcegepant hydrochloride (Synonyms: BIBN-4096 hydrochloride; BIBN4096BS hydrochloride)
CAS586368-06-1
FormulaC38H47Br2N9O5.HCl
MW906.11
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Olcegepant hydrochloride (BIBN-4096 hydrochloride) is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide 1 (CGRP1) receptor with IC50 of 0.03 nM and with a Ki of 14.4 pM for human CGRP.

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Olcegepant (Synonyms: BIBN-4096; BIBN 4096BS)
History
Olcegepant hydrochloride (Synonyms: BIBN-4096 hydrochloride; BIBN4096BS hydrochloride)
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