SB408124 HCl
SB-408124 Hydrochloride
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Product Overview
Product Name SB-408124 Hydrochloride
CAS1431697-90-3
FormulaC19H18F2N4O·HCl
MW392.83 | 356.38(free)
AppearanceWhite to gray powder
Storage condition4°C, sealed storage, away from moisture
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Product details

SB-408124 Hydrochloride is a selective non-peptide orexin receptor 1 (OX1) receptor antagonist with Kis of 57 nM and 27 nM in whole cell and membrane, respectively. SB-408124 Hydrochloride exhibits 50-fold selectivity over OX2 receptor.


Related
H-89 Dihydrochloride | H 89 2HCl
History
SB-408124 Hydrochloride