3-(1-甲基-1H-吲哚-3-基)-4-(1-(1-(2-吡啶甲基)-4-哌啶基)-1H-吲哚-3-基)-1H-吡咯-2,5-二酮;恩扎妥林
Enzastaurin (Synonyms: LY317615)
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Product Overview
Product Name Enzastaurin (Synonyms: LY317615)
CAS170364-57-5
FormulaC32 H29 N5 O2
MW515.60
MDLMFCD11040980
AppearancePink to red powder
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Product details

Enzastaurin (LY317615) is an effective inhibitor of PKCβ with an IC50 value of 6 nM. Enzastaurin shows 6-20 times greater selectivity for PKCβ compared to PKCα, PKCγ, and PKCε.

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History
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