6-氯-9-[(4-甲氧基-3,5-二甲基-2-吡啶基)甲基]-9H-嘌呤-2-胺
BIIB021 (Synonyms: CNF2024;BIIB-021;BIIB 021)
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Product Name BIIB021 (Synonyms: CNF2024;BIIB-021;BIIB 021)
CAS848695-25-0
FormulaC14H15ClN6O
MW318.76
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BIIB021 (CNF2024) is an orally active, fully synthetic inhibitor of HSP90 with a Ki and an EC50 of 1.7 nM and 38 nM, respectively.
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