9-羟基利培酮; 帕潘立酮
Paliperidone (Synonyms: 9-Hydroxyrisperidone)
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250 mg 500 mg 1 g
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$250.00
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$300.00
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Product Overview
Product Name Paliperidone (Synonyms: 9-Hydroxyrisperidone)
CAS144598-75-4
FormulaC23H27FN4O3
MW426.48
AppearanceWhite to off-white powder
Storage condition Dry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years).
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Paliperidone, the main active metabolite of Risperidone, is a potent serotonin-2A and dopamine-2 receptor antagonist, used in the treatment of schizophrenia.
Paliperidone (9-Hydroxyrisperidone), the major active metabolite of Risperidone, is a dopamine D2 antagonist and 5-HT2A antagonist. Paliperidone is also active as an antagonist at α1 and α2 adrenergic receptors and H1-histaminergic receptors. Paliperidone, a antipsychotic agent, shows efficacy against schizophrenia.

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