BIX02188
BIX02188
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Product Name BIX02188
CAS334949-59-6
FormulaC25H24N4O2
MW412.49
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BIX02188 is a potent MEK5-selective inhibitor with an IC50 of 4.3 nM. BIX02188 inhibits ERK5 catalytic activity, with an IC50 of 810 nM.

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History
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D-Isoleucine (Synonyms: (R)-Isoleucine)
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Tenofovir (Synonyms:GS 1278; PMPA)
BIX02188
Fondaparinux sodium (Synonyms: Fondaparin sodium; SR-90107A)
Lartesertib (Synonyms: M4076; ATM Inhibitor-5)
(R)-Roscovitine (Synonyms: Seliciclib; CYC202,细胞周期蛋白B激酶抑制剂;塞利西利)
Batoprotafib (Synonyms: TNO155); (3S,4S)-8-(6-Amino-5-((2-amino-3-chloropyridin-4-yl)thio)pyrazin-2-yl)-3-methyl-2-oxa-8-azaspiro[4.5]decan-4-amine
Safinamide (FCE 26743; EMD 1195686)