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Ponatinib (Synonyms: AP24534)
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Product Overview
Product Name Ponatinib (Synonyms: AP24534)
CAS943319-70-8
FormulaC29H27F3N6O
MW532.56
Melting point >160 °C
AppearanceLight yellow to yellow powder
Storage conditionDry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years).
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Ponatinib (AP24534) is an orally active multi-targeted kinase inhibitor with IC50s of 0.37 nM, 1.1 nM, 1.5 nM, 2.2 nM, and 5.4 nM for AblPDGFRαVEGFR2FGFR1, and Src, respectively.
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History
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