格佐匹韦 | 格拉瑞韦
Grazoprevir (Synonyms: MK-5172)
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Product Name Grazoprevir (Synonyms: MK-5172)
CAS1350514-68-9
FormulaC38H50N6O9S
MW766.90
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Grazoprevir (MK-5172) is a selective inhibitor of Hepatitis C virus NS3/4a protease with broad activity across genotypes and resistant variants, with Kis of 0.01 nM (gt1b), 0.01 nM (gt1a), 0.08 nM (gt2a), 0.15 nM (gt2b), 0.90 nM (gt3a), respectively. Grazoprevir inhibits SARS-CoV-2 3CLpro activity.
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