1-(4-(3-氨基-1H-吲唑-4-基)苯基)-3-(2-氟-5-甲基苯基)脲; 利尼伐尼
Linifanib(ABT-869; AL-39324; RG3635)
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3-5days
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$66.00
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Product Availability
3-5days
Price
$96.00
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Product Availability
3-5days
Price
$166.00
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Product Overview
Product Name Linifanib(ABT-869; AL-39324; RG3635)
CAS796967-16-3
FormulaC21H18FN5O
MW375.40
MDLMFCD11840918
AppearanceWhite to gray powder
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Product details

Linifanib (formerly RG3635, ABT869, AL39324) is an orally bioavailable and ATP-competitive inhibitor of multiple kinases (e.g. VEGFR/PDGFR) with potential antitumor activity. Its IC50 values are 4 nM, 3 nM, 3 nM/4 nM, and 66 nM for KDR, CSF-1R, Flt-1/3, and PDGFRβ, respectively. Linifanib has strong antitumor efficaciousness in vivo and outstanding anti-proliferative activity in vitro.

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History
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