2-[(2-氯-4-碘苯基)氨基]-N-(环丙基甲氧基)-3,4-二氟-苯甲酰胺
PD184352(Synonyms: CI-1040)
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3-5days
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$100.00
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Product Availability
3-5days
Price
$160.00
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Product Availability
3-5days
Price
$290.00
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Product Overview
Product Name PD184352(Synonyms: CI-1040)
CAS212631-79-3
FormulaC17H14ClF2 IN2O2
MW478.66
MDLMFCD02683961
AppearanceWhite to off-white powder
Storage condition Dry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years).
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Product details

PD184352 (PD-184352; CI-1040), an analog of benzhydroxamate, is an orally bioactive, specific, allosteric/non-ATP competitive MEK1/2 inhibitor with potential anticancer activity. In cell-based assays, it inhibits MEK1/2 with IC50 values of 17 nM and exhibits a 100-fold preference for MEK1/2 over MEK5. In mouse xenograft models, it exhibits strong in vitro anti-proliferative activity and significant in vivo antitumor efficacy.

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