阿帕替尼
Apatinib | Apatinib Free base | YN968D1| Rivoceranib
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1 mg 5 mg
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$148.00
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$288.00
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Product Overview
Product Name Apatinib | Apatinib Free base | YN968D1| Rivoceranib
CAS811803-05-1
FormulaC24H23N5O
MW397.47
Storage conditionStore in a dry and dark sealed container, short-term (weeks to months) storage at 0-4 ℃, long-term (months to years) storage at -20 ℃.
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Product details

Apatinib (Rivoceranib, YN968D1) is a potent inhibitor of the VEGF signaling pathway with IC50 values of 1 nM, 13 nM, 429 nM and 530 nM for VEGFR-2, Ret (c-Ret), c-Kit and c-Src, respectively. Apatinib induces both autophagy and apoptosis.


Related
Apatinib Mesylate
History
Belinostat (Synonyms: PXD101; PX105684; NSC726630; PX-105684)
Phenformin Hydrochloride (Synonyms: Phenformin HCl; Phenethylbiguanide hydrochloride; NSC-756501)
Epothilone B (Synonyms: EPO 906; Patupilone)
Lasmiditan (Synonyms: COL-144; LY573144)
Apatinib | Apatinib Free base | YN968D1| Rivoceranib
tert-butyl 2-(3-(2-aMino-2-oxoacetyl)-1-benzyl-2-ethyl-1H-indol-4-yloxy)acetate
Atropine hydrobromide | Tropine tropate hydrobromide | DL-Hyoscyamine hydrobromide
(R)-Bicalutamide
Erlotinib Hydrochloride (Synonyms: Erlotinib HCl; CP-358774 hydrochloride; NSC 718781 hydrochloride; OSI-774 hydrochloride; OSI-774 HCl)
(S)-N-((4-(((1,4-dioxan-2-yl)methyl)amino)-3-nitrophenyl)sulfonyl)-2-((1H-pyrrolo[2,3-b]pyridin-5-yl)oxy)-4-(4-((6-(4-chlorophenyl)spiro[3.5]non-6-en-7-yl)methyl)piperazin-1-yl)benzamide