阿帕替尼
Apatinib | Apatinib Free base | YN968D1| Rivoceranib
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1 mg 5 mg
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$148.00
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In-stock
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$288.00
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Product Overview
Product Name Apatinib | Apatinib Free base | YN968D1| Rivoceranib
CAS811803-05-1
FormulaC24H23N5O
MW397.47
Storage conditionStore in a dry and dark sealed container, short-term (weeks to months) storage at 0-4 ℃, long-term (months to years) storage at -20 ℃.
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Product details

Apatinib (Rivoceranib, YN968D1) is a potent inhibitor of the VEGF signaling pathway with IC50 values of 1 nM, 13 nM, 429 nM and 530 nM for VEGFR-2, Ret (c-Ret), c-Kit and c-Src, respectively. Apatinib induces both autophagy and apoptosis.


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