阿帕替尼甲磺酸盐
Apatinib Mesylate
ChemLeader
Catalog No:
CAS No.:
MDLNo:
Formula:
MW:
Size
1 mg 5 mg
Product Availability
3-5days
Price
$148.00
Member price
Product Availability
3-5days
Price
$288.00
Member price
Quantity
- +
Product Overview
Product Name Apatinib Mesylate
CAS1218779-75-9
FormulaC24H23N5O · CH4O3S
MW493.58 | 397.48(free)
Security information
Product details

 

Apatinib mesylate (YN968D1, Rivoceranib) is a potent inhibitor of the VEGF signaling pathway with IC50 values of 1 nM, 13 nM, 429 nM and 530 nM for VEGFR-2, Ret (c-Ret), c-Kit and c-Src, respectively. Apatinib mesylate induces both autophagy and apoptosis.


Related
Apatinib | Apatinib Free base | YN968D1| Rivoceranib
History
Apatinib Mesylate
Fmoc-Val-Thr[PSI(Me,Me)Pro]-OH
DL-Glutamic Acid Monohydrate
Fmoc-6-Ahx-OH/Fmoc-ε-Acp-OH
Secretin | swine
Tegoprazan | CJ-12420 | IN-A001 | K-CAB | LXI-15028 | RQ-00000004
KAAD-Cyclopamine (Synonyms: Cyclopamine-KAAD;3-Keto-N-aminoethyl-N’-aminocaproyldihydrocinnamoyl Cyclopamine)
CX-5461 dihydrochloride
Atazanavir Sulfate (Synonyms: BMS-232632 Sulfate)
Miglustat Hydrochloride (N-Butyldeoxynojirimycin Hydrochloride; NB-DNJ hydrochloride; OGT918 hydrochloride)