赛乐西帕 | 司来帕格
Selexipag (Synonyms: NS-304; ACT-293987)
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Product Availability
3-5days
Price
$100.00
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Product Availability
3-5days
Price
$125.00
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Product Availability
3-5days
Price
$200.00
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Product Overview
Product Name Selexipag (Synonyms: NS-304; ACT-293987)
CAS475086-01-2
FormulaC26H32N4O4S
MW496.62
Appearance White to yellow powder
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Product details

Selexipag, also known as ACT-293987 and NS-304, is a a first-in-class orally available selective non-prostanoid IP receptor agonist, which is currently in development by Actelion as a treatment of pulmonary arterial hypertension. Selexipag and its active metabolite, ACT-333679, are agonists at the prostacyclin receptor, which leads to vasodilation in the pulmonary circulation.

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History
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