INS018-055 (TNIK&MAP4K4-IN-2)
Rentosertib (Synonyms: INS018-055;ISM001-055;TNIK&MAP4K4-IN-2)
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Product Name Rentosertib (Synonyms: INS018-055;ISM001-055;TNIK&MAP4K4-IN-2)
CAS2828567-39-9
FormulaC27H30FN7O
MW487.57
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Rentosertib (INS018 055) (compound 112) is the orally active TNIK and MAP4K4 inhibitor with IC50 values of 12-120, 12-120 nM, respectively.
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