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Osilodrostat (Synonyms: LCI699)
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1 mg 5 mg 10 mg
Product Availability
3-5days
Price
$100.00
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Product Availability
3-5days
Price
$165.00
Member price
Product Availability
3-5days
Price
$288.00
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Product Overview
Product Name Osilodrostat (Synonyms: LCI699)
CAS928134-65-0
FormulaC13H10FN3
MW227.24
AppearanceWhite to yellow pwder
Storage conditionDry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years).
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Product details

Osilodrostat, also known as LCI699, is a potent inhibitor of 11β-hydroxylase, the enzyme which catalyzes the final step of cortisol synthesis. LCI699 may thus be a potential new treatment for all forms of Cushing's syndrome. Current evidence indicates that the novel aldosterone inhibitor LCI699 is an effective and well-tolerated antihypertensive agent that lowers plasma aldosterone concentration and produces a mild ACTH-stimulated cortisol response suppressive effect.
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