特戈拉赞
Tegoprazan | CJ-12420 | IN-A001 | K-CAB | LXI-15028 | RQ-00000004
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Product Name Tegoprazan | CJ-12420 | IN-A001 | K-CAB | LXI-15028 | RQ-00000004
CAS942195-55-3
FormulaC20H19F2N3O3
MW387.38
AppearanceOff-white to light yellow powder
Storage conditionDry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years).
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Tegoprazan (CJ-12420, IN-A001, K-CAB, LXI-15028, RQ-00000004) is a novel potent and highly selective inhibitor of gastric H+/K+-ATPase with IC50s ranging from 0.29 μM to 0.52 μM for porcine, canine, and human H+/K+-ATPases in vitro, respectively.

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History
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