BIX-01294盐酸盐水合物
BIX-01294 hydrochloride hydrate
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Product Name BIX-01294 hydrochloride hydrate
CAS1808255-64-2
FormulaC28H38N6O2.3ClH.xH2O
MW
Storage conditionStore in a dry and dark sealed container, short-term (weeks to months) storage at 0-4 ℃, long-term (months to years) storage at -20 ℃.
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BIX-01294 hydrochloride hydrate is a histone-lysine methyltransferase (HMTase) inhibitor, which selective inhibits the G9aHMTase with IC50 of 1.7 μM, reduces histone-3 lysine (9) methylation (H3K9me), induces autophagy and apoptosis in human glioma cells.


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