PT100
Talabostat (Synonyms: Val-boroPro; PT100)
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Product Overview
Product Name Talabostat (Synonyms: Val-boroPro; PT100)
CAS149682-77-9
FormulaC9H19BN2O3
MW214.07
Storage conditionStore in a dry and dark sealed container, short-term (weeks to months) storage at 0-4 ℃, long-term (months to years) storage at -20 ℃.
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Product details

Talabostat (Val-boroPro, PT-100) is a dipeptidyl peptidase inhibitor with IC50 values of <4 nM, 4 nM, 11 nM, 310 nM, 560 nM and 390 nM for DPP-IV, DPP8, DPP9, QPP, FAP and PEP respectively. It has antineoplastic and hematopoiesis- stimulating activities.


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History
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