(3R,4R) 替凡替尼 (ARQ 197), 肝细胞生长因子受体抑制剂 | 替万替尼
Tivantinib | ARQ-197
ChemLeader
Catalog No:
CAS No.:
MDLNo:
Formula:
MW:
Size
Quantity
- +
Product Overview
Product Name Tivantinib | ARQ-197
CAS905854-02-6
FormulaC23H19N3O2
MW369.42
AppearanceLight brown to brown powder
Security information
Product details

Tivantinib is the first non-ATP-competitive c-Met inhibitor with Ki of 0.355 μM in a cell-free assay, little activity to Ron, and no inhibition to EGFR, InsR, PDGFRα or FGFR1/4. Tivantinib (ARQ 197) induces a G2/M arrest and apoptosis.


Related
Sorry, no related items
History
Valrubicin | AD-32
Ciclesonide (RPR251526)
Anti-Human RSV Monoclonal Antibody(Motavizumab)
Vapaliximab
Benralizumab (Anti-IL-5Ra/ CD125)
Anti-Human IL-23 Monoclonal Antibody(Guselkumab)
Thunberginol C
Taxiphyllin
Tivantinib | ARQ-197
Rhodionin | Herbacetin-7-O-glucorhamnoside