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Rosiglitazone potassium | BRL 49653 potassium
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Product Name Rosiglitazone potassium | BRL 49653 potassium
CAS316371-84-3
FormulaC18H18N3O3S • K
MW395.5
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Rosiglitazone (BRL 49653) potassium is an orally active selective PPARγ agonist (EC50: 60 nM, Kd: 40 nM). Rosiglitazone potassium is a TRPC5 activator (EC50: 30 μM) and TRPM3 inhibitor. Rosiglitazone potassium can be used in the research of obesity and diabetes, senescence, ovarian cancer.


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History
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AZD3965