甲磺酸达布非龙
Darbufelone mesilate | CI-1004 mesylate
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Product Overview
Product Name Darbufelone mesilate | CI-1004 mesylate
CAS139340-56-0
FormulaC18H24N2O2S·CH4O3S
MW428.57 | 332.46 (free)
AppearanceWhite to light yellow powder
Storage condition4°C, sealed storage, away from moisture and light
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Product details

Darbufelone mesylate (CI-1004 mesylate) is a dual inhibitor of cellular PGF and LTB4 production. Darbufelone potently inhibits PGHS-2 (IC50 = 0.19 μM) but is much less potent with PGHS-1 (IC50= 20 μM).


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