磷酸鲁索替尼 | 磷酸芦可替尼 | 磷酸鲁索利替尼
Ruxolitinib phosphate (Synonyms: INCB018424 phosphate;INCB-018424 phosphate)
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Product Overview
Product Name Ruxolitinib phosphate (Synonyms: INCB018424 phosphate;INCB-018424 phosphate)
CAS1092939-17-7
FormulaC17H18N6·H3PO4
MW404.36 | 306.37(free)
AppearanceWhite to gray powder
Storage condition4°C, sealed storage, away from moisture
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Product details

Ruxolitinib phosphate (INCB018424 phosphate) is a potent JAK1/2 inhibitor with IC50s of 3.3 nM/2.8 nM, respectively, showing more than 130-fold selectivity over JAK3.


Related
Ruxolitinib sulfate | INCB018424 sulfate
Ruxolitinib (Synonyms: Ruxolitinib Free base; INCB18424;(R)-Ruxolitinib)
History
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