鲁索替尼硫酸盐 | 鲁索利替尼硫酸盐
Ruxolitinib sulfate | INCB018424 sulfate
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Product Overview
Product Name Ruxolitinib sulfate | INCB018424 sulfate
CAS1092939-16-6
FormulaC17H18N6 · H2SO4
MW404.44 | 306.37(free)
AppearanceOff-white to gray powder
Storage condition4°C, sealed storage, away from moisture
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Product details

Ruxolitinib sulfate (INCB018424 sulfate) is the first potent, selective JAK1/2 inhibitor to enter the clinic with IC50s of 3.3 nM/2.8 nM, and has > 130-fold selectivity for JAK1/2 versus JAK3.


Related
Ruxolitinib phosphate (Synonyms: INCB018424 phosphate;INCB-018424 phosphate)
Ruxolitinib (Synonyms: Ruxolitinib Free base; INCB18424;(R)-Ruxolitinib)
History
Goserelin Acetate
Calcitonin Acetate(Salmon); Salcitonin Acetate
Atazanavir (Synonyms: Atazanavir Base; BMS-232632)
Dapsone (DDS)
Ruxolitinib sulfate | INCB018424 sulfate
EDTA disodium (Synonyms: Ethylenediamine tetraacetic acid disodium salt)
Tariquidar dihydrochloride | XR9576 dihydrochloride
Tolcapone | Ro 40-7592
Ramiprilat (Synonyms: HOE 498 diacid; Ramipril diacid)
Lusutrombopag (Synonyms: S-888711)