鲁索替尼硫酸盐 | 鲁索利替尼硫酸盐
Ruxolitinib sulfate | INCB018424 sulfate
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Product Overview
Product Name Ruxolitinib sulfate | INCB018424 sulfate
CAS1092939-16-6
FormulaC17H18N6 · H2SO4
MW404.44 | 306.37(free)
AppearanceOff-white to gray powder
Storage condition4°C, sealed storage, away from moisture
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Product details

Ruxolitinib sulfate (INCB018424 sulfate) is the first potent, selective JAK1/2 inhibitor to enter the clinic with IC50s of 3.3 nM/2.8 nM, and has > 130-fold selectivity for JAK1/2 versus JAK3.


Related
Ruxolitinib phosphate| INCB-018424 phosphate
Ruxolitinib | INCB018424 | Ruxolitinib Free base | (R)-Ruxolitinib
History
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