8-(4-(1-氨基环丁基)苯基)-9-苯基-[1,2,4]三唑并[3,4-f][1,6]萘啶-3(2H)-酮二盐酸盐
MK-2206 dihydrochloride | MK-2206 ·2HCl
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Product Overview
Product Name MK-2206 dihydrochloride | MK-2206 ·2HCl
CAS1032350-13-2
FormulaC25H23N5O· 2HCl
MW482.40
MDLMFCD14584463
AppearanceYellow powder
Storage condition 4°C, sealed storage, away from moisture
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Product details

MK-2206 dihydrochloride (MK-2206 (2HCl)) is an orally active, BBB-penetrated allosteric AKT inhibitor with IC50s of 5 nM, 12 nM, and 65 nM for AKT1AKT2, and AKT3, respectively. MK-2206 dihydrochloride induces autophagy.


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History
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