4-((2R,3S,4S,5R)-3-(3,4-二氟-2-甲氧基苯基)-4,5-二甲基-5-(三氟甲基)四氢呋喃-2-甲酰胺)吡啶-2-甲酰胺
Suzetrigine (Synonyms: VX-548)
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1 mg 5 mg
Product Availability
3-5 days
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$466.00
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Product Availability
3-5 days
Price
$1066.00
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Product Overview
Product Name Suzetrigine (Synonyms: VX-548)
CAS2649467-58-1
FormulaC21H20F5N3O4
MW473.39
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Product details

Suzetrigine (VX-548) is a selective NaV1.8 inhibitor with oral bioavailability, acting as a potent analgesic. It targets the sodium channel protein type 10 subunit alpha, playing a key role in pain transmission. This drug candidate shows promise in acute pain management post-abdominoplasty and bunionectomy, presenting as a non-opioid analgesic option.


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History
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