N-(5-(4-氰基苯基)-1H-吡咯并[2,3-b]吡啶-3-基)吡啶-3-甲酰胺
Pim1/AKK1-IN-1 (Synonyms: LKB1/AAK1 dual inhibitor)
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Product Name Pim1/AKK1-IN-1 (Synonyms: LKB1/AAK1 dual inhibitor)
CAS1093222-27-5
FormulaC20H13N5O
MW339.35
MDLMFCD15528944
AppearanceWhite to gray powder
Storage conditionStore short-term at 0-4°C or long-term at -20°C in a dry, dark place.
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Product details

 Pim1/AKK1-IN-1 is a potent multi-kinase inhibitor with Kd values of 35 nM/53 nM/75 nM/380 nM for Pim1/AKK1/MST2/LKB1 respectively, and it also inhibits MPSK1 and TNIK.


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History
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