6-(3-氨基苄基)-4-甲基-2-(甲基亚磺酰基)-4H-噻吩并[2',3':4,5]吡咯并[2,3-d]哒嗪-5(6H)-酮
TEPP-46 (Synonyms: ML-265)
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3-5 days
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Product Overview
Product Name TEPP-46 (Synonyms: ML-265)
CAS1221186-53-3
FormulaC17H16N4O2S2
MW372.46
MDLMFCD23160747
AppearanceWhite to light yellow powder
Storage conditionStore short-term at 0-4°C or long-term at -20°C in a dry, dark place.
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Product details

TEPP-46, also known as ML265, is a potent and selective PKM2 activator with an AC50 of 92 nM, exhibiting high selectivity over PKM1, PKR, and PKL.

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History
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