(E)-N-[4-[(3-氯-4-氟苯基)氨基]-3-氰基-7-乙氧基-6-喹啉基]-4-(二甲基氨基)-2-丁烯酰胺; 培利替尼; 贝利替尼
Pelitinib (Synonyms: EKB-569; WAY-EKB 569)
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Product Overview
Product Name Pelitinib (Synonyms: EKB-569; WAY-EKB 569)
CAS257933-82-7
FormulaC24H23ClFN5O2
MW467.92
MDLMFCD09837868
AppearanceWhite to off-white powder
Storage conditionStore short-term at 0-4°C or long-term at -20°C in a dry, dark place.
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Product details

Pelitinib (EKB-569) is a potent, irreversible EGFR inhibitor with an IC50 of 38.5 nM, displaying selectivity over Src, MEK/ERK, and ErbB2 with respective IC50s of 282 nM, 800 nM, and 1255 nM.

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History
Teniposide (Synonyms: VM26;NSC 122819;VM-26)
Efavirenz (Synonyms: DMP 266; EFV; L-743726; DMP-266)
GSK583
Pelitinib (Synonyms: EKB-569; WAY-EKB 569)
Tariquidar dimesylate | XR9576 dimesylate
Vicriviroc maleate (Synonyms: SCH-417690 maleate ; SCH-D maleate; 维立韦罗马来酸盐)
StreptoMycin sulfate | NSC 14083
Telaprevir | VX-950 | LY-570310 | MP-424
Orantinib | SU 6668 | TSU-68
Tozasertib(VX-680;MK-0457)