Product Name | Elacestrant (Synonyms: RAD1901) |
---|---|
CAS | 722533-56-4 |
Formula | C30H38N2O2 |
MW | 458.63 |
MDL | MFCD30532693 |
Appearance | White to off-white powder |
Storage condition | 4°C, sealed storage, away from moisture and light |
Elacestrant (RAD1901) is a potent oral SERD with IC50s of 48 nM for ERα and 870 nM for ERβ. It effectively inhibits the growth of ER+ breast cancer cell lines both in vitro and in vivo, showcasing its significant bioactivity in targeting estrogen receptor pathways crucial for cancer cell proliferation.
© Copyright 2015-2021 Chemleader Biomedical Co., Ltd. All Rights Reserved.
沪ICP备15046197号-4
沪公网安备31011502007856号
Designed by Kuanersoft