| Product Name | Elacestrant (Synonyms: RAD1901) |
|---|---|
| CAS | 722533-56-4 |
| Formula | C30H38N2O2 |
| MW | 458.63 |
| MDL | MFCD30532693 |
| Appearance | White to off-white powder |
| Storage condition | 4°C, sealed storage, away from moisture and light |
Elacestrant (RAD1901) is a potent oral SERD with IC50s of 48 nM for ERα and 870 nM for ERβ. It effectively inhibits the growth of ER+ breast cancer cell lines both in vitro and in vivo, showcasing its significant bioactivity in targeting estrogen receptor pathways crucial for cancer cell proliferation.
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