SB-742457 (GSK-742457; RVT-101; Intepirdine)
Intepirdine (Synonyms: SB-742457; GSK-742457; RVT-101)
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Product Name Intepirdine (Synonyms: SB-742457; GSK-742457; RVT-101)
CAS607742-69-8
FormulaC19H19N3O2S
MW353.44
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Intepirdine (SB742457) is a highly selective 5-HT6 receptor antagonist with pKi of 9.63; exhibits >100-fold selectivity over other receptors.
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