DPCPX (Synonyms: PD 116948);CAS: DPCPX (Synonyms: PD 116948)

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Product Overview

Product Name	DPCPX (Synonyms: PD 116948)
CAS	102146-07-6
Formula	C16H24N4O2
MW	304.39
MDL	MFCD00055117
Appearance	White to off-white powder
Storage condition	Store short-term at 0-4°C or long-term at -20°C in a dry, dark place.

Product details

DPCPX (PD 116948), derived from xanthine, is an exceptionally potent and selective inhibitor of the Adenosine A1 receptor. It shows a high affinity with a Ki value of 0.46 nM for binding to A1 receptors, as determined by 3H-CHA binding assays in rat whole brain membrane preparations.

Related literature

PD 116,948, a Highly Selective A1 Adenosine Receptor Antagonist.

PMID: 3807648 DOI: 10.1016/0024-3205(87)90369-9

DPCPX, a selective adenosine A1 receptor antagonist, enhances the antidepressant-like effects of imipramine, escitalopram, and reboxetine in mice behavioral tests

PMID: 30094458 PMCID: PMC6208968 DOI: 10.1007/s00210-018-1551-z

The Adenosine A1 Receptor Antagonist DPCPX Inhibits Tumor Progression via the ERK/JNK Pathway in Renal Cell Carcinoma

PMID: 28950257 DOI: 10.1159/000481557

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History

CL3115

DPCPX (Synonyms: PD 116948)

102146-07-6 98+%

DPCPX (Synonyms: PD 116948)

Chemical safety data sheet(MSDS)