Ketanserin tartrate | R41468 tartrate

Size	Availability	Price(USD)	VIP Price (USD)	Quantity
50 mg	In-stock	$56.00	Visible after login	- +
100 mg	In-stock	$76.00	Visible after login	- +
250 mg	In-stock	$156.00	Visible after login	- +
500 mg	In-stock	$226.00	Visible after login	- +
1 g	In-stock	$368.00	Visible after login	- +
2 g	3-5days	$636.00	Visible after login	- +

Size

Availability

Price(USD)

VIP Price (USD)

Quantity

50 mg

In-stock

$56.00

Visible after login

- +

100 mg

In-stock

$76.00

Visible after login

- +

250 mg

In-stock

$156.00

Visible after login

- +

500 mg

In-stock

$226.00

Visible after login

- +

1 g

In-stock

$368.00

Visible after login

- +

2 g

3-5days

$636.00

Visible after login

- +

Product Overview

Product Name	Ketanserin tartrate \| R41468 tartrate
CAS	83846-83-7
Formula	C26H28FN3O9
MW	545.51
Appearance	White to off-white powder
Storage condition	Dry, dark and at 0 - 4 ℃ for short term (days to weeks) or -20 ℃ for long term (months to years).

Product details

Ketanserin (R41468) tartrate is a selective 5-HT2 receptor antagonist. Ketanserin tartrate also blocks hERG current (I_hERG) in a concentration-dependent manner (IC₅₀=0.11 μM).

Related literature

Investigation of cyclooxygenase and signaling pathways involved in human platelet aggregation mediated by synergistic interaction of various agonists.

PMID: 26185418 PMCID: PMC4500629 DOI: 10.2147/DDDT.S84335

The 5-HT2 antagonist Ketanserin is an open channel blocker of human cardiac ether-à-go-go-related gene (hERG) potassium channels.

PMID: 18574455 PMCID: PMC2567890 DOI: 10.1038/bjp.2008.261

Antiserotonergic properties of terguride in blood vessels, platelets, and valvular interstitial cells.

PMID: 22049464 DOI: 10.1124/jpet.111.187906

Serotonin regulates brain-derived neurotrophic factor expression in select brain regions during acute psychological stress.

PMID: 27857753 PMCID: PMC5090852 DOI: 10.4103/1673-5374.191222

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History

CL2348A