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Size	Availability	Price(USD)	VIP Price (USD)	Quantity
1 mg	3-5 days	$156.00	Visible after login	- +
2 mg	3-5 days	$246.00	Visible after login	- +
5 mg	3-5 days	$456.00	Visible after login	- +

Size

Availability

Price(USD)

VIP Price (USD)

Quantity

1 mg

3-5 days

$156.00

Visible after login

- +

2 mg

3-5 days

$246.00

Visible after login

- +

5 mg

3-5 days

$456.00

Visible after login

- +

Product Overview

Product Name	Elacestrant (Synonyms: RAD1901)
CAS	722533-56-4
Formula	C30H38N2O2
MW	458.63
MDL	MFCD30532693
Appearance	White to off-white powder
Storage condition	4°C, sealed storage, away from moisture and light

Product details

Elacestrant (RAD1901) is a potent oral SERD with IC50s of 48 nM for ERα and 870 nM for ERβ. It effectively inhibits the growth of ER+ breast cancer cell lines both in vitro and in vivo, showcasing its significant bioactivity in targeting estrogen receptor pathways crucial for cancer cell proliferation.

Related literature

RAD1901: a novel, orally bioavailable selective estrogen receptor degrader that demonstrates antitumor activity in breast cancer xenograft models.

PMID: 26164151 PMCID: PMC4560273 DOI: 10.1097/CAD.0000000000000271

Elacestrant (RAD1901), a Selective Estrogen Receptor Degrader (SERD), Has Antitumor Activity in Multiple ER+ Breast Cancer Patient-derived Xenograft Models.

PMID: 28473534 DOI: 10.1158/1078-0432.CCR-16-2561

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History

CL3146

Elacestrant (Synonyms: RAD1901)

722533-56-4 98+%

Elacestrant (Synonyms: RAD1901)

Chemical safety data sheet(MSDS)